PDB Information

PDB5NGB
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceMus musculus
Primary Citation
Identification of a Potent Phosphoinositide 3-Kinase Pan Inhibitor Displaying a Strategic Carboxylic Acid Group and Development of Its Prodrugs.
Pirali, T., Ciraolo, E., Aprile, S., Massarotti, A., Berndt, A., Griglio, A., Serafini, M., Mercalli, V., Landoni, C., Campa, C.C., Margaria, J.P., Silva, R.L., Grosa, G., Sorba, G., Williams, R., Hirsch, E., Tron, G.C.
ChemMedChem
HeaderTransferase
Released2017-03-17
Resolution2.900
CATH Insert Date14 Nov, 2017

PDB Images (7)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Chopped

CATH Domains (5)

Domain ID Date inserted into CATH Superfamily CATH Status
5ngbA01 10 Dec, 2017 1.25.40.70 Assigned
5ngbA02 10 Dec, 2017 3.10.20.90 Assigned
5ngbA03 10 Dec, 2017 2.60.40.150 Assigned
5ngbA04 10 Dec, 2017 3.30.1010.10 Assigned
5ngbA05 10 Dec, 2017 1.10.1070.11 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O35904 PK3CD_MOUSE Mus musculus Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform