Discovery of Pyrazolo[1,5-a]pyrimidine B-Cell Lymphoma 6 (BCL6) Binders and Optimization to High Affinity Macrocyclic Inhibitors.
McCoull, W., Abrams, R.D., Anderson, E., Blades, K., Barton, P., Box, M., Burgess, J., Byth, K., Cao, Q., Chuaqui, C., Carbajo, R.J., Cheung, T., Code, E., Ferguson, A.D., Fillery, S., Fuller, N.O., Gangl, E., Gao, N., Grist, M., Hargreaves, D., Howard, M.R., Hu, J., Kemmitt, P.D., Nelson, J.E., O'Connell, N., Prince, D.B., Raubo, P., Rawlins, P.B., Robb, G.R., Shi, J., Waring, M.J., Whittaker, D., Wylot, M., Zhu, X.
J. Med. Chem.