PDB Information

PDB5M7M
MethodX-RAY DIFFRACTION
Host OrganismHomo sapiens
Gene SourceHomo sapiens
Primary Citation
Discovery, Structure-Activity Relationship, and Binding Mode of an Imidazo[1,2-a]pyridine Series of Autotaxin Inhibitors.
Joncour, A., Desroy, N., Housseman, C., Bock, X., Bienvenu, N., Cherel, L., Labeguere, V., Peixoto, C., Annoot, D., Lepissier, L., Heiermann, J., Hengeveld, W.J., Pilzak, G., Monjardet, A., Wakselman, E., Roncoroni, V., Le Tallec, S., Galien, R., David, C., Vandervoort, N., Christophe, T., Conrath, K., Jans, M., Wohlkonig, A., Soror, S., Steyaert, J., Touitou, R., Fleury, D., Vercheval, L., Mollat, P., Triballeau, N., van der Aar, E., Brys, R., Heckmann, B.
J. Med. Chem.
HeaderHydrolase
Released2016-10-28
Resolution2.700
CATH Insert Date14 Nov, 2017

PDB Images (2)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 14 Nov, 2017 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q13822 ENPP2_HUMAN Homo sapiens Ectonucleotide pyrophosphatase/phosphodiesterase family member 2