PDB Information

PDB5LWN
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Selective JAK3 Inhibitors with a Covalent Reversible Binding Mode Targeting a New Induced Fit Binding Pocket.
Forster, M., Chaikuad, A., Bauer, S.M., Holstein, J., Robers, M.B., Corona, C.R., Gehringer, M., Pfaffenrot, E., Ghoreschi, K., Knapp, S., Laufer, S.A.
Cell Chem Biol
HeaderTransferase
Released2016-09-18
Resolution1.600
CATH Insert Date06 Nov, 2016

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Nov, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5lwnA01 10 Nov, 2016 3.30.200.20 Assigned
5lwnA02 10 Nov, 2016 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P52333 JAK3_HUMAN Homo sapiens Tyrosine-protein kinase JAK3