PDB Information

PDB5LQQ
MethodX-RAY DIFFRACTION
Host OrganismHomo sapiens
Gene SourceRattus norvegicus
Primary Citation
Structure-Activity Relationships of Small Molecule Autotaxin Inhibitors with a Discrete Binding Mode.
Miller, L.M., Keune, W.J., Castagna, D., Young, L.C., Duffy, E.L., Potjewyd, F., Salgado-Polo, F., Engel Garcia, P., Semaan, D., Pritchard, J.M., Perrakis, A., Macdonald, S.J., Jamieson, C., Watson, A.J.
J. Med. Chem.
HeaderHydrolase
Released2016-08-17
Resolution2.400
CATH Insert Date08 Jan, 2017

PDB Images (6)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 09 Jan, 2017 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5lqqA01 19 Jan, 2017 Holding pen
5lqqA02 19 Jan, 2017 4.10.410.20 Assigned
5lqqA03 19 Jan, 2017 3.40.720.10 Assigned
5lqqA04 19 Jan, 2017 3.40.570.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q64610 ENPP2_RAT Rattus norvegicus Ectonucleotide pyrophosphatase/phosphodiesterase family member 2