PDB Information

PDB5KKR
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Small molecule stabilization of the KSR inactive state antagonizes oncogenic Ras signalling.
Dhawan, N.S., Scopton, A.P., Dar, A.C.
Nature
HeaderTransferase
Released2016-06-22
Resolution3.510
CATH Insert Date09 Oct, 2016

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
B 10 Oct, 2016 Chopped
C 10 Oct, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5kkrB01 13 Oct, 2016 3.30.200.20 Assigned
5kkrB02 13 Oct, 2016 1.10.510.10 Assigned
5kkrC01 13 Oct, 2016 3.30.200.20 Assigned
5kkrC02 13 Oct, 2016 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P29678 MP2K1_RABIT Oryctolagus cuniculus Dual specificity mitogen-activated protein kinase kinase 1
Q6VAB6 KSR2_HUMAN Homo sapiens Kinase suppressor of Ras 2