PDB Information

PDB5IGM
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Promiscuous targeting of bromodomains by bromosporine identifies BET proteins as master regulators of primary transcription response in leukemia.
Picaud, S., Leonards, K., Lambert, J.P., Dovey, O., Wells, C., Fedorov, O., Monteiro, O., Fujisawa, T., Wang, C.Y., Lingard, H., Tallant, C., Nikbin, N., Guetzoyan, L., Ingham, R., Ley, S.V., Brennan, P., Muller, S., Samsonova, A., Gingras, A.C., Schwaller, J., Vassiliou, G., Knapp, S., Filippakopoulos, P.
Sci Adv
HeaderTranscription
Released2016-02-28
Resolution1.600
CATH Insert Date06 Nov, 2016

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 07 Nov, 2016 Chopped
B 07 Nov, 2016 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
5igmA00 10 Nov, 2016 1.20.920.10 Assigned
5igmB00 10 Nov, 2016 1.20.920.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9H8M2 BRD9_HUMAN Homo sapiens Bromodomain-containing protein 9
Q9H8M2 BRD9_HUMAN Homo sapiens Bromodomain-containing protein 9