PDB Information

PDB5HLN
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Inhibitors of Glycogen Synthase Kinase 3 with Exquisite Kinome-Wide Selectivity and Their Functional Effects.
Wagner, F.F., Bishop, J.A., Gale, J.P., Shi, X., Walk, M., Ketterman, J., Patnaik, D., Barker, D., Walpita, D., Campbell, A.J., Nguyen, S., Lewis, M., Ross, L., Weiwer, M., An, W.F., Germain, A.R., Nag, P.P., Metkar, S., Kaya, T., Dandapani, S., Olson, D.E., Barbe, A.L., Lazzaro, F., Sacher, J.R., Cheah, J.H., Fei, D., Perez, J., Munoz, B., Palmer, M., Stegmaier, K., Schreiber, S.L., Scolnick, E., Zhang, Y.L., Haggarty, S.J., Holson, E.B., Pan, J.Q.
Acs Chem.Biol.
HeaderTransferase/Transferase Inhibitor
Released2016-01-15
Resolution3.100
CATH Insert Date05 Jun, 2016

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 06 Jun, 2016 Chopped
B 06 Jun, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5hlnA01 16 Jul, 2016 3.30.200.20 Assigned
5hlnA02 16 Jul, 2016 1.10.510.10 Assigned
5hlnB01 17 Jul, 2016 3.30.200.20 Assigned
5hlnB02 17 Jul, 2016 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P49841 GSK3B_HUMAN Homo sapiens Glycogen synthase kinase-3 beta
P49841 GSK3B_HUMAN Homo sapiens Glycogen synthase kinase-3 beta