PDB Information

PDB5GGZ
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Novel Tetrahydropyrido[4,3-d]pyrimidines as Potent Inhibitors of Chaperone Heat Shock Protein 90
Jiang, F., Wang, H.J., Jin, Y.H., Zhang, Q., Wang, Z.H., Jia, J.M., Liu, F., Wang, L., Bao, Q.C., Li, D.D., You, Q.D., Xu, X.L.
J. Med. Chem.
HeaderChaperone/Chaperone Inhibitor
Released2016-06-16
Resolution2.020
CATH Insert Date07 May, 2017

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 08 May, 2017 Chopped
B 08 May, 2017 Chopped
C 08 May, 2017 Chopped
D 08 May, 2017 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5ggzA00 12 May, 2017 3.30.565.10 Assigned
5ggzB00 12 May, 2017 3.30.565.10 Assigned
5ggzC00 12 May, 2017 3.30.565.10 Assigned
5ggzD00 12 May, 2017 3.30.565.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P07900 HS90A_HUMAN Homo sapiens Heat shock protein HSP 90-alpha
P07900 HS90A_HUMAN Homo sapiens Heat shock protein HSP 90-alpha
P07900 HS90A_HUMAN Homo sapiens Heat shock protein HSP 90-alpha
P07900 HS90A_HUMAN Homo sapiens Heat shock protein HSP 90-alpha