PDB 5g4r

PDB Information

PDB5G4R
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Gsk6853, a Chemical Probe for Inhibition of the Brpf1 Bromodomain.
Bamborough, P., Barnett, H.A., Becher, I., Bird, M.J., Chung, C., Craggs, P.D., Demont, E.H., Diallo, H., Fallon, D.J., Gordon, L.J., Grandi, P., Hobbs, C.I., Hooper-Greenhill, E., Jones, E.J., Law, R.P., Le Gall, A., Lugo, D., Michon, A., Mitchell, D.J., Prinjha, R.K., Sheppard, R.J., Watson, A.J.B., Watson, R.J.
Acs Med.Chem.Lett.
HeaderTranscription
Released2016-05-16
Resolution1.960
CATH Insert Date24 Jul, 2016

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 25 Jul, 2016 Chopped
B 25 Jul, 2016 Chopped
C 25 Jul, 2016 Chopped
D 25 Jul, 2016 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5g4rA00 01 Sep, 2016 1.20.920.10 Assigned
5g4rB00 01 Sep, 2016 1.20.920.10 Assigned
5g4rC00 01 Sep, 2016 1.20.920.10 Assigned
5g4rD00 01 Sep, 2016 1.20.920.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P55201 BRPF1_HUMAN Homo sapiens Peregrin
P55201 BRPF1_HUMAN Homo sapiens Peregrin
P55201 BRPF1_HUMAN Homo sapiens Peregrin
P55201 BRPF1_HUMAN Homo sapiens Peregrin