PDB Information

PDB5FHO
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceRattus norvegicus
Primary Citation
Tweaking Subtype Selectivity and Agonist Efficacy at (S)-2-Amino-3-(3-hydroxy-5-methyl-isoxazol-4-yl)propionic acid (AMPA) Receptors in a Small Series of BnTetAMPA Analogues.
Wang, S.Y., Larsen, Y., Navarrete, C.V., Jensen, A.A., Nielsen, B., Al-Musaed, A., Frydenvang, K., Kastrup, J.S., Pickering, D.S., Clausen, R.P.
J.Med.Chem.
HeaderMembrane Protein
Released2015-12-22
Resolution2.300
CATH Insert Date10 Apr, 2016

PDB Images (13)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Chopped
B 11 Apr, 2016 Chopped
C 11 Apr, 2016 Chopped
D 11 Apr, 2016 Chopped

CATH Domains (8)

Domain ID Date inserted into CATH Superfamily CATH Status
5fhoA01 11 May, 2016 3.40.190.10 Assigned
5fhoA02 11 May, 2016 3.40.190.10 Assigned
5fhoB01 11 May, 2016 3.40.190.10 Assigned
5fhoB02 11 May, 2016 3.40.190.10 Assigned
5fhoC01 11 May, 2016 3.40.190.10 Assigned
5fhoC02 11 May, 2016 3.40.190.10 Assigned
5fhoD01 11 May, 2016 3.40.190.10 Assigned
5fhoD02 11 May, 2016 3.40.190.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P19491 GRIA2_RAT Rattus norvegicus Glutamate receptor 2
P19491 GRIA2_RAT Rattus norvegicus Glutamate receptor 2
P19491 GRIA2_RAT Rattus norvegicus Glutamate receptor 2
P19491 GRIA2_RAT Rattus norvegicus Glutamate receptor 2