PDB 5f95
PDB Information
PDB | 5F95 |
Method | X-RAY DIFFRACTION |
Host Organism | unidentified baculovirus |
Gene Source | Homo sapiens |
Primary Citation | Discovery of Isonicotinamides as Highly Selective, Brain Penetrable, and Orally Active Glycogen Synthase Kinase-3 Inhibitors.
J.Med.Chem.
|
Header | Transferase/Transferase Inhibitor |
Released | 2015-12-09 |
Resolution | 2.530 |
CATH Insert Date | 10 Apr, 2016 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 11 Apr, 2016 | Chopped |
B | 11 Apr, 2016 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5f95A01 | 10 May, 2016 | 3.30.200.20 | Assigned |
5f95A02 | 10 May, 2016 | 1.10.510.10 | Assigned |
5f95B01 | 10 May, 2016 | 3.30.200.20 | Assigned |
5f95B02 | 10 May, 2016 | 1.10.510.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P49841 | GSK3B_HUMAN | Homo sapiens | Glycogen synthase kinase-3 beta |
P49841 | GSK3B_HUMAN | Homo sapiens | Glycogen synthase kinase-3 beta |