PDB Information

PDB5EAP
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-Based Optimization of a Small Molecule Antagonist of the Interaction Between WD Repeat-Containing Protein 5 (WDR5) and Mixed-Lineage Leukemia 1 (MLL1).
Getlik, M., Smil, D., Zepeda-Velazquez, C., Bolshan, Y., Poda, G., Wu, H., Dong, A., Kuznetsova, E., Marcellus, R., Senisterra, G., Dombrovski, L., Hajian, T., Kiyota, T., Schapira, M., Arrowsmith, C.H., Brown, P.J., Vedadi, M., Al-Awar, R.
J. Med. Chem.
HeaderTranscription/Transcription Inhibitor
Released2015-10-16
Resolution1.730
CATH Insert Date15 Nov, 2015

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 16 Nov, 2015 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
5eapA00 24 Nov, 2015 2.130.10.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P61964 WDR5_HUMAN Homo sapiens WD repeat-containing protein 5