PDB 5eap
PDB Information
PDB | 5EAP |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Structure-Based Optimization of a Small Molecule Antagonist of the Interaction Between WD Repeat-Containing Protein 5 (WDR5) and Mixed-Lineage Leukemia 1 (MLL1).
J. Med. Chem.
|
Header | Transcription/Transcription Inhibitor |
Released | 2015-10-16 |
Resolution | 1.730 |
CATH Insert Date | 15 Nov, 2015 |
PDB Images (3)
PDB Prints
PDB Chains (1)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 16 Nov, 2015 | Chopped |
CATH Domains (1)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5eapA00 | 24 Nov, 2015 | 2.130.10.10 | Assigned |
UniProtKB Entries (1)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P61964 | WDR5_HUMAN | Homo sapiens | WD repeat-containing protein 5 |