PDB 5eak

PDB Information

PDB5EAK
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
Optimization of microtubule affinity regulating kinase (MARK) inhibitors with improved physical properties.
Sloman, D.L., Noucti, N., Altman, M.D., Chen, D., Mislak, A.C., Szewczak, A., Hayashi, M., Warren, L., Dellovade, T., Wu, Z., Marcus, J., Walker, D., Su, H.P., Edavettal, S.C., Munshi, S., Hutton, M., Nuthall, H., Stanton, M.G.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2015-10-16
Resolution2.800
CATH Insert Date10 Apr, 2016

PDB Images (3)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 11 Apr, 2016 Holding pen
B 11 Apr, 2016 Holding pen

CATH Domains (0)

Domain ID Date inserted into CATH Superfamily CATH Status

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q7KZI7 MARK2_HUMAN Homo sapiens Serine/threonine-protein kinase MARK2
Q7KZI7 MARK2_HUMAN Homo sapiens Serine/threonine-protein kinase MARK2