PDB Information

PDB5CTP
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli BL21(DE3)
Gene SourceHomo sapiens
Primary Citation
A fragment-based approach leading to the discovery of a novel binding site and the selective CK2 inhibitor CAM4066.
De Fusco, C., Brear, P., Iegre, J., Georgiou, K.H., Sore, H.F., Hyvonen, M., Spring, D.R.
Bioorg. Med. Chem.
HeaderTransferase
Released2015-07-24
Resolution2.030
CATH Insert Date08 Jan, 2017

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 09 Jan, 2017 Chopped
B 09 Jan, 2017 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
5ctpA01 18 Jan, 2017 1.10.510.10 Assigned
5ctpA02 18 Jan, 2017 3.30.200.20 Assigned
5ctpB01 18 Jan, 2017 1.10.510.10 Assigned
5ctpB02 18 Jan, 2017 3.30.200.20 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P68400 CSK21_HUMAN Homo sapiens Casein kinase II subunit alpha
P68400 CSK21_HUMAN Homo sapiens Casein kinase II subunit alpha