PDB 5coi
PDB Information
PDB | 5COI |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli BL21(DE3) |
Gene Source | Homo sapiens |
Primary Citation | Discovery of Benzo[cd]indol-2(1H)-ones as Potent and Specific BET Bromodomain Inhibitors: Structure-Based Virtual Screening, Optimization, and Biological Evaluation
J.Med.Chem.
|
Header | Signaling Protein/Inhibitor |
Released | 2015-07-20 |
Resolution | 1.620 |
CATH Insert Date | 10 Apr, 2016 |
PDB Images (3)
PDB Prints
PDB Chains (1)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 11 Apr, 2016 | Chopped |
CATH Domains (1)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
5coiA01 | 05 May, 2016 | 1.20.920.10 | Assigned |
UniProtKB Entries (1)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
O60885 | BRD4_HUMAN | Homo sapiens | Bromodomain-containing protein 4 |