PDB Information

PDB5A4E
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Probing the ATP-Binding Pocket of Protein Kinase Dyrk1A with Benzothiazole Fragment Molecules
Rothweiler, U., Stensen, W., Brandsdal, B.O., Isaksson, J., Leeson, F.A., Eugh, R.A., Mjoen Svendsen, J.S.
J.Med.Chem.
HeaderTransferase
Released2015-06-08
Resolution2.680
CATH Insert Date10 Jul, 2016

PDB Images (12)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 11 Jul, 2016 Chopped
B 11 Jul, 2016 Chopped
C 11 Jul, 2016 Chopped
D 11 Jul, 2016 Chopped

CATH Domains (7)

Domain ID Date inserted into CATH Superfamily CATH Status
5a4eA01 30 Nov, 2016 3.30.200.20 Assigned
5a4eA02 30 Nov, 2016 1.10.510.10 Assigned
5a4eB01 13 Jul, 2016 3.30.200.20 Assigned
5a4eB02 13 Jul, 2016 1.10.510.10 Assigned
5a4eC00 29 Nov, 2016 1.10.510.10 Assigned
5a4eD01 13 Jul, 2016 3.30.200.20 Assigned
5a4eD02 13 Jul, 2016 1.10.510.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A