PDB Information

PDB4ZOM
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of novel pyrazole-containing benzamides as potent ROR gamma inverse agonists.
Wang, T., Banerjee, D., Bohnert, T., Chao, J., Enyedy, I., Fontenot, J., Guertin, K., Jones, H., Lin, E.Y., Marcotte, D., Talreja, T., Van Vloten, K.
Bioorg.Med.Chem.Lett.
HeaderTranscription
Released2015-05-06
Resolution2.270
CATH Insert Date28 Jun, 2015

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped
C 29 Jun, 2015 Chopped
D 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4zomA00 27 Jul, 2015 1.10.565.10 Assigned
4zomB00 27 Jul, 2015 1.10.565.10 Assigned
4zomC00 27 Jul, 2015 1.10.565.10 Assigned
4zomD00 27 Jul, 2015 1.10.565.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P51449 RORG_HUMAN Homo sapiens Nuclear receptor ROR-gamma
P51449 RORG_HUMAN Homo sapiens Nuclear receptor ROR-gamma
P51449 RORG_HUMAN Homo sapiens Nuclear receptor ROR-gamma
P51449 RORG_HUMAN Homo sapiens Nuclear receptor ROR-gamma