PDB Information

PDB4ZJR
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of biaryl carboxylamides as potent ROR gamma inverse agonists.
Chao, J., Enyedy, I., Van Vloten, K., Marcotte, D., Guertin, K., Hutchings, R., Powell, N., Jones, H., Bohnert, T., Peng, C.C., Silvian, L., Hong, V.S., Little, K., Banerjee, D., Peng, L., Taveras, A., Viney, J.L., Fontenot, J.
Bioorg.Med.Chem.Lett.
HeaderTranscription
Released2015-04-29
Resolution2.700
CATH Insert Date28 Jun, 2015

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped
C 29 Jun, 2015 Chopped
D 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4zjrA00 27 Jul, 2015 1.10.565.10 Assigned
4zjrB00 27 Jul, 2015 1.10.565.10 Assigned
4zjrC00 27 Jul, 2015 1.10.565.10 Assigned
4zjrD00 27 Jul, 2015 1.10.565.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P51449 RORG_HUMAN Homo sapiens Nuclear receptor ROR-gamma
P51449 RORG_HUMAN Homo sapiens Nuclear receptor ROR-gamma
P51449 RORG_HUMAN Homo sapiens Nuclear receptor ROR-gamma
P51449 RORG_HUMAN Homo sapiens Nuclear receptor ROR-gamma