PDB Information

PDB4X3R
MethodX-RAY DIFFRACTION
Host OrganismDrosophila melanogaster
Gene SourceHomo sapiens
Primary Citation
Design of highly potent urea-based, exosite-binding inhibitors selective for glutamate carboxypeptidase II.
Tykvart, J., Schimer, J., Jancarik, A., Barinkova, J., Navratil, V., Starkova, J., Sramkova, K., Konvalinka, J., Majer, P., Sacha, P.
J.Med.Chem.
HeaderHydrolase
Released2014-12-01
Resolution1.860
CATH Insert Date25 Oct, 2015

PDB Images (5)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 26 Oct, 2015 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
4x3rA01 04 Jan, 2017 3.40.630.10 Assigned
4x3rA02 04 Jan, 2017 3.50.30.30 Assigned
4x3rA03 04 Jan, 2017 1.20.930.40 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q04609 FOLH1_HUMAN Homo sapiens Glutamate carboxypeptidase 2