PDB Information

PDB4UY1
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Discovery of a Novel Pyrazole Series of Group X Secreted Phospholipase A2 Inhibitor (Spla2X) Via Fragment Based Virtual Screening
Chen, H., Knerr, L., Akerud, T., Hallberg, K., Bodin, C., Oster, L., Rohman, M., Osterlund, K., Beisel, H.G., Olsson, T., Brengdhal, J., Sandmark, J.
Bioorg.Med.Chem.Lett.
HeaderHydrolase
Released2014-08-28
Resolution2.200
CATH Insert Date26 Oct, 2014

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 27 Oct, 2014 Chopped
B 27 Oct, 2014 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4uy1A00 02 Nov, 2014 1.20.90.10 Assigned
4uy1B00 02 Nov, 2014 1.20.90.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O15496 PA2GX_HUMAN Homo sapiens Group 10 secretory phospholipase A2
O15496 PA2GX_HUMAN Homo sapiens Group 10 secretory phospholipase A2