PDB Information

PDB4RVM
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Mitigation of Acetylcholine Esterase Activity in the 1,7-Diazacarbazole Series of Inhibitors of Checkpoint Kinase 1.
Gazzard, L., Williams, K., Chen, H., Axford, L., Blackwood, E., Burton, B., Chapman, K., Crackett, P., Drobnick, J., Ellwood, C., Epler, J., Flagella, M., Gancia, E., Gill, M., Goodacre, S., Halladay, J., Hewitt, J., Hunt, H., Kintz, S., Lyssikatos, J., Macleod, C., Major, S., Medard, G., Narukulla, R., Ramiscal, J., Schmidt, S., Seward, E., Wiesmann, C., Wu, P., Yee, S., Yen, I., Malek, S.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2014-11-26
Resolution1.860
CATH Insert Date28 Jun, 2015

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4rvmA01 10 Jul, 2015 3.30.200.20 Assigned
4rvmA02 10 Jul, 2015 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O14757 CHK1_HUMAN Homo sapiens Serine/threonine-protein kinase Chk1