PDB Information

PDB4R6T
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourcePlasmodium falciparum 3D7
Primary Citation
Two-Pronged Attack: Dual Inhibition of Plasmodium falciparum M1 and M17 Metalloaminopeptidases by a Novel Series of Hydroxamic Acid-Based Inhibitors.
Mistry, S.N., Drinkwater, N., Ruggeri, C., Sivaraman, K.K., Loganathan, S., Fletcher, S., Drag, M., Paiardini, A., Avery, V.M., Scammells, P.J., McGowan, S.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2014-08-26
Resolution2.600
CATH Insert Date09 Nov, 2014

PDB Images (37)

PDB Prints

PDB Chains (12)

Chain ID Date inserted into CATH CATH Status
A 10 Nov, 2014 Chopped
B 10 Nov, 2014 Chopped
C 10 Nov, 2014 Chopped
D 10 Nov, 2014 Chopped
E 10 Nov, 2014 Chopped
F 10 Nov, 2014 Chopped
G 10 Nov, 2014 Chopped
H 10 Nov, 2014 Chopped
I 10 Nov, 2014 Chopped
J 10 Nov, 2014 Chopped
K 10 Nov, 2014 Chopped
L 10 Nov, 2014 Chopped

CATH Domains (24)

Domain ID Date inserted into CATH Superfamily CATH Status
4r6tA01 14 Nov, 2014 3.40.220.10 Assigned
4r6tA02 14 Nov, 2014 3.40.630.10 Assigned
4r6tB01 14 Nov, 2014 3.40.220.10 Assigned
4r6tB02 14 Nov, 2014 3.40.630.10 Assigned
4r6tC01 13 Nov, 2014 3.40.220.10 Assigned
4r6tC02 13 Nov, 2014 3.40.630.10 Assigned
4r6tD01 14 Nov, 2014 3.40.220.10 Assigned
4r6tD02 14 Nov, 2014 3.40.630.10 Assigned
4r6tE01 13 Nov, 2014 3.40.220.10 Assigned
4r6tE02 13 Nov, 2014 3.40.630.10 Assigned
4r6tF01 14 Nov, 2014 3.40.220.10 Assigned
4r6tF02 14 Nov, 2014 3.40.630.10 Assigned
4r6tG01 13 Nov, 2014 3.40.220.10 Assigned
4r6tG02 13 Nov, 2014 3.40.630.10 Assigned
4r6tH01 14 Nov, 2014 3.40.220.10 Assigned
4r6tH02 14 Nov, 2014 3.40.630.10 Assigned
4r6tI01 14 Nov, 2014 3.40.220.10 Assigned
4r6tI02 14 Nov, 2014 3.40.630.10 Assigned
4r6tJ01 13 Nov, 2014 3.40.220.10 Assigned
4r6tJ02 13 Nov, 2014 3.40.630.10 Assigned
4r6tK01 12 Nov, 2014 3.40.220.10 Assigned
4r6tK02 12 Nov, 2014 3.40.630.10 Assigned
4r6tL01 14 Nov, 2014 3.40.220.10 Assigned
4r6tL02 14 Nov, 2014 3.40.630.10 Assigned

UniProtKB Entries (12)

Accession Gene ID Taxon Description
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase
Q8IL11 Q8IL11_PLAF7 Plasmodium falciparum 3D7 M17 leucyl aminopeptidase