PDB Information

PDB4Q0L
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery and characterization of novel selective inhibitors of carbonic anhydrase IX.
Dudutiene, V., Matuliene, J., Smirnov, A., Timm, D.D., Zubriene, A., Baranauskiene, L., Morkunaite, V., Smirnoviene, J., Michailoviene, V., Juozapaitiene, V., Mickeviciute, A., Kazokaite, J., Baksyte, S., Kasiliauskaite, A., Jachno, J., Revuckiene, J., Kisonaite, M., Pilipuityte, V., Ivanauskaite, E., Milinaviciute, G., Smirnovas, V., Petrikaite, V., Kairys, V., Petrauskas, V., Norvaisas, P., Linge, D., Gibieza, P., Capkauskaite, E., Zaksauskas, A., Kazlauskas, E., Manakova, E., Grazulis, S., Ladbury, J.E., Matulis, D.
J.Med.Chem.
HeaderLyase/Lyase Inhibitor
Released2014-04-02
Resolution2.000
CATH Insert Date28 Jun, 2015

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped
C 29 Jun, 2015 Chopped
D 29 Jun, 2015 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4q0lA00 09 Jul, 2015 3.10.200.10 Assigned
4q0lB00 10 Jul, 2015 3.10.200.10 Assigned
4q0lC00 09 Jul, 2015 3.10.200.10 Assigned
4q0lD00 10 Jul, 2015 3.10.200.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
O43570 CAH12_HUMAN Homo sapiens Carbonic anhydrase 12
O43570 CAH12_HUMAN Homo sapiens Carbonic anhydrase 12
O43570 CAH12_HUMAN Homo sapiens Carbonic anhydrase 12
O43570 CAH12_HUMAN Homo sapiens Carbonic anhydrase 12