PDB Information

PDB4PXS
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery and Structure-Guided Optimization of Diarylmethanesulfonamide Disruptors of GK-GKRP Binding.
Pennington, L.D., Bartberger, M.D., Croghan, M.D., Andrews, K.L., Ashton, K.S., Bourbeau, M.P., Chen, J., Chmait, S., Cupples, R., Fotsch, C.
To be Published
HeaderTransferase/Transferase Inhibitor
Released2014-03-24
Resolution2.600
CATH Insert Date28 Jun, 2015

PDB Images (9)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 29 Jun, 2015 Chopped
B 29 Jun, 2015 Chopped

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
4pxsA01 10 Jul, 2015 3.40.50.10490 Assigned
4pxsA02 10 Jul, 2015 Holding pen
4pxsA03 10 Jul, 2015 Holding pen
4pxsB01 10 Jul, 2015 3.40.50.10490 Assigned
4pxsB02 10 Jul, 2015 Holding pen
4pxsB03 10 Jul, 2015 Holding pen

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein
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