PDB Information

PDB4PJV
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structural basis for the inhibition of poly(ADP-ribose) polymerases 1 and 2 by BMN 673, a potent inhibitor derived from dihydropyridophthalazinone.
Aoyagi-Scharber, M., Gardberg, A.S., Yip, B.K., Wang, B., Shen, Y., Fitzpatrick, P.A.
Acta Crystallogr.,Sect.F
HeaderTransferase/Transferase Inhibitor
Released2014-05-12
Resolution2.500
CATH Insert Date05 Oct, 2014

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 06 Oct, 2014 Chopped
B 06 Oct, 2014 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4pjvA01 07 Oct, 2014 1.20.142.10 Assigned
4pjvA02 07 Oct, 2014 3.90.228.10 Assigned
4pjvB01 08 Oct, 2014 1.20.142.10 Assigned
4pjvB02 08 Oct, 2014 3.90.228.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q9UGN5 PARP2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase 2
Q9UGN5 PARP2_HUMAN Homo sapiens Poly [ADP-ribose] polymerase 2