PDB 4pf3

PDB Information

PDB4PF3
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of 6-[5-(4-fluorophenyl)-3-methyl-pyrazol-4-yl]-benzoxazin-3-one derivatives as novel selective nonsteroidal mineralocorticoid receptor antagonists
Hasui, T., Ohyabu, N., Ohra, T., Fuji, K., Sugimoto, T., Fujimoto, J., Asano, K., Oosawa, M., Shiotani, S., Nishigaki, N., Kusumoto, K., Matsui, H., Mizukami, A., Habuka, N., Sogabe, S., Endo, S., Ono, M., Siedem, C.S., Tang, T.P., Gauthier, C., De Meese, L.A., Boyd, S.A., Fukumoto, S.
Bioorg.Med.Chem.
HeaderTranscription/Transcription Inhibitor
Released2014-04-28
Resolution1.100
CATH Insert Date07 Dec, 2014

PDB Images (3)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Dec, 2014 Chopped

CATH Domains (1)

Domain ID Date inserted into CATH Superfamily CATH Status
4pf3A00 28 Dec, 2014 1.10.565.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P08235 MCR_HUMAN Homo sapiens Mineralocorticoid receptor