PDB Information

PDB4ONA
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceToxoplasma gondii
Primary Citation
Potent and selective inhibitors of CDPK1 from T. gondii and C. parvum based on a 5-aminopyrazole-4-carboxamide scaffold.
Zhang, Z., Ojo, K.K., Vidadala, R., Huang, W., Geiger, J.A., Scheele, S., Choi, R., Reid, M.C., Keyloun, K.R., Rivas, K., Siddaramaiah, L.K., Comess, K.M., Robinson, K.P., Merta, P.J., Kifle, L., Hol, W.G., Parsons, M., Merritt, E.A., Maly, D.J., Verlinde, C.L., Van Voorhis, W.C., Fan, E.
ACS Med Chem Lett
HeaderTransferase/Transferase Inhibitor
Released2014-01-28
Resolution2.400
CATH Insert Date23 Mar, 2014

PDB Images (5)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 24 Mar, 2014 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
4onaA01 25 Apr, 2014 3.30.200.20 Assigned
4onaA02 25 Apr, 2014 1.10.510.10 Assigned
4onaA03 25 Apr, 2014 Holding pen

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9BJF5 Q9BJF5_TOXGO Toxoplasma gondii Calmodulin-domain protein kinase 1