PDB 4nie
PDB Information
PDB | 4NIE |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Discovery of Tertiary Amine and Indole Derivatives as Potent ROR gamma t Inverse Agonists.
Acs Med.Chem.Lett.
|
Header | Transcription/Agonist |
Released | 2013-11-06 |
Resolution | 2.010 |
CATH Insert Date | 15 Dec, 2013 |
PDB Images (7)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 16 Dec, 2013 | Chopped |
B | 16 Dec, 2013 | Chopped |
C | 16 Dec, 2013 | Rejected |
D | 16 Dec, 2013 | Rejected |
CATH Domains (2)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4nieA00 | 20 Dec, 2013 | 1.10.565.10 | Assigned |
4nieB00 | 20 Dec, 2013 | 1.10.565.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q15596 | NCOA2_HUMAN | Homo sapiens | Nuclear receptor coactivator 2 |
Q15596 | NCOA2_HUMAN | Homo sapiens | Nuclear receptor coactivator 2 |
P51449 | RORG_HUMAN | Homo sapiens | Nuclear receptor ROR-gamma |
P51449 | RORG_HUMAN | Homo sapiens | Nuclear receptor ROR-gamma |