PDB Information

PDB4MSU
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Small Molecule Disruptors of the Glucokinase-Glucokinase Regulatory Protein Interaction: 1. Discovery of a Novel Tool Compound for in Vivo Proof-of-Concept.
Ashton, K.S., Andrews, K.L., Bryan, M.C., Chen, J., Chen, K., Chen, M., Chmait, S., Croghan, M., Cupples, R., Fotsch, C., Helmering, J., Jordan, S.R., Kurzeja, R.J., Michelsen, K., Pennington, L.D., Poon, S.F., Sivits, G., Van, G., Vonderfecht, S.L., Wahl, R.C., Zhang, J., Lloyd, D.J., Hale, C., St Jean, D.J.
J.Med.Chem.
HeaderSugar Binding Protein
Released2013-09-18
Resolution2.500
CATH Insert Date16 Mar, 2014

PDB Images (9)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 17 Mar, 2014 Chopped
B 17 Mar, 2014 Chopped

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
4msuA01 25 Apr, 2014 3.40.50.10490 Assigned
4msuA02 25 Apr, 2014 Holding pen
4msuA03 25 Apr, 2014 Holding pen
4msuB01 17 Apr, 2014 3.40.50.10490 Assigned
4msuB02 17 Apr, 2014 Holding pen
4msuB03 17 Apr, 2014 Holding pen

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein
Q14397 GCKR_HUMAN Homo sapiens Glucokinase regulatory protein