PDB 4mr3

PDB Links
Overview

PDB Information

PDB	4MR3
Method	X-RAY DIFFRACTION
Host Organism	Escherichia coli
Gene Source	Homo sapiens
Primary Citation	RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain. Picaud, S., Wells, C., Felletar, I., Brotherton, D., Martin, S., Savitsky, P., Diez-Dacal, B., Philpott, M., Bountra, C., Lingard, H., Fedorov, O., Muller, S., Brennan, P.E., Knapp, S., Filippakopoulos, P. Proc.Natl.Acad.Sci.USA
Header	Transcription/Transcription Inhibitor
Released	2013-09-17
Resolution	1.680
CATH Insert Date	01 Dec, 2013

PDB Images (3)

Image of CATH 4mr3

4mr3

PDB 4mr3

Image of CATH 4mr3A

4mr3A

PDB Chain 4mr3A

Image of CATH 4mr3A01

4mr3A01

CATH Domain 4mr3A01

PDB Prints

PDB Chains (1)

Chain ID	Date inserted into CATH	CATH Status
A	02 Dec, 2013	Chopped

CATH Domains (1)

Domain ID	Date inserted into CATH	Superfamily	CATH Status
4mr3A01	04 Dec, 2013	1.20.920.10	Assigned

UniProtKB Entries (1)

Accession	Gene ID	Taxon	Description
O60885	BRD4_HUMAN	Homo sapiens	Bromodomain-containing protein 4