PDB Information

PDB4M84
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceToxoplasma gondii
Primary Citation
Potent and selective inhibitors of CDPK1 from T. gondii and C. parvum based on a 5-aminopyrazole-4-carboxamide scaffold.
Zhang, Z., Ojo, K.K., Vidadala, R., Huang, W., Geiger, J.A., Scheele, S., Choi, R., Reid, M.C., Keyloun, K.R., Rivas, K., Siddaramaiah, L.K., Comess, K.M., Robinson, K.P., Merta, P.J., Kifle, L., Hol, W.G., Parsons, M., Merritt, E.A., Maly, D.J., Verlinde, C.L., Van Voorhis, W.C., Fan, E.
ACS Med Chem Lett
HeaderTransferase/Transferase Inhibitor
Released2013-08-12
Resolution2.000
CATH Insert Date06 Oct, 2013

PDB Images (5)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 07 Oct, 2013 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
4m84A01 10 Oct, 2013 3.30.200.20 Assigned
4m84A02 10 Oct, 2013 1.10.510.10 Assigned
4m84A03 10 Oct, 2013 Holding pen

UniProtKB Entries (1)

Accession Gene ID Taxon Description
Q9BJF5 Q9BJF5_TOXGO Toxoplasma gondii Calmodulin-domain protein kinase 1