PDB Information

PDB4L7F
MethodX-RAY DIFFRACTION
Host Organism
Gene SourceHomo sapiens
Primary Citation
Hit-to-lead optimization and kinase selectivity of imidazo[1,2-a]quinoxalin-4-amine derived JNK1 inhibitors.
Li, B., Cociorva, O.M., Nomanbhoy, T., Weissig, H., Li, Q., Nakamura, K., Liyanage, M., Zhang, M.C., Shih, A.Y., Aban, A., Hu, Y., Cajica, J., Pham, L., Kozarich, J.W., Shreder, K.R.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Inhibitor
Released2013-06-13
Resolution1.950
CATH Insert Date01 Sep, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 02 Sep, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4l7fA01 10 Sep, 2013 3.30.200.20 Assigned
4l7fA02 10 Sep, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P45983 MK08_HUMAN Homo sapiens Mitogen-activated protein kinase 8