PDB Information

PDB4KB9
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHuman immunodeficiency virus 1
Primary Citation
Highly Potent HIV-1 Protease Inhibitors with Novel Tricyclic P2 Ligands: Design, Synthesis, and Protein-Ligand X-ray Studies.
Ghosh, A.K., Parham, G.L., Martyr, C.D., Nyalapatla, P.R., Osswald, H.L., Agniswamy, J., Wang, Y.F., Amano, M., Weber, I.T., Mitsuya, H.
J.Med.Chem.
HeaderHydrolase/Hydrolase Inhibitor
Released2013-04-23
Resolution1.290
CATH Insert Date22 Sep, 2013

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 23 Sep, 2013 Chopped
B 23 Sep, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4kb9A00 25 Sep, 2013 2.40.70.10 Assigned
4kb9B00 25 Sep, 2013 2.40.70.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q7SSI0 Q7SSI0_9HIV1 Human immunodeficiency virus 1 Protease
Q7SSI0 Q7SSI0_9HIV1 Human immunodeficiency virus 1 Protease