PDB Information

PDB4JPG
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of 2-((1H-benzo[d]imidazol-1-yl)methyl)-4H-pyrido[1,2-a]pyrimidin-4-ones as novel PKM2 activators.
Guo, C., Linton, A., Jalaie, M., Kephart, S., Ornelas, M., Pairish, M., Greasley, S., Richardson, P., Maegley, K., Hickey, M., Li, J., Wu, X., Ji, X., Xie, Z.
Bioorg.Med.Chem.Lett.
HeaderTransferase/Transferase Activator
Released2013-03-19
Resolution2.330
CATH Insert Date07 Jul, 2013

PDB Images (17)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped
B 08 Jul, 2013 Chopped
C 08 Jul, 2013 Chopped
D 08 Jul, 2013 Chopped

CATH Domains (12)

Domain ID Date inserted into CATH Superfamily CATH Status
4jpgA01 09 Aug, 2013 3.40.1380.20 Assigned
4jpgA02 09 Aug, 2013 3.20.20.60 Assigned
4jpgA03 09 Aug, 2013 2.40.33.10 Assigned
4jpgB01 09 Aug, 2013 3.40.1380.20 Assigned
4jpgB02 09 Aug, 2013 3.20.20.60 Assigned
4jpgB03 09 Aug, 2013 2.40.33.10 Assigned
4jpgC01 09 Aug, 2013 3.40.1380.20 Assigned
4jpgC02 09 Aug, 2013 3.20.20.60 Assigned
4jpgC03 09 Aug, 2013 2.40.33.10 Assigned
4jpgD01 09 Aug, 2013 3.40.1380.20 Assigned
4jpgD02 09 Aug, 2013 3.20.20.60 Assigned
4jpgD03 09 Aug, 2013 2.40.33.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
P14618 KPYM_HUMAN Homo sapiens Pyruvate kinase PKM
P14618 KPYM_HUMAN Homo sapiens Pyruvate kinase PKM
P14618 KPYM_HUMAN Homo sapiens Pyruvate kinase PKM
P14618 KPYM_HUMAN Homo sapiens Pyruvate kinase PKM