(R)-PFI-2 is a potent and selective inhibitor of SETD7 methyltransferase activity in cells.
Barsyte-Lovejoy, D., Li, F., Oudhoff, M.J., Tatlock, J.H., Dong, A., Zeng, H., Wu, H., Freeman, S.A., Schapira, M., Senisterra, G.A., Kuznetsova, E., Marcellus, R., Allali-Hassani, A., Kennedy, S., Lambert, J.P., Couzens, A.L., Aman, A., Gingras, A.C., Al-Awar, R., Fish, P.V., Gerstenberger, B.S., Roberts, L., Benn, C.L., Grimley, R.L., Braam, M.J., Rossi, F.M., Sudol, M., Brown, P.J., Bunnage, M.E., Owen, D.R., Zaph, C., Vedadi, M., Arrowsmith, C.H.
Proc.Natl.Acad.Sci.USA
