PDB Information

PDB4HGT
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Structure-Based Design of Potent and Selective CK1 gamma Inhibitors.
Huang, H., Acquaviva, L., Berry, V., Bregman, H., Chakka, N., O'Connor, A., DiMauro, E.F., Dovey, J., Epstein, O., Grubinska, B., Goldstein, J., Gunaydin, H., Hua, Z., Huang, X., Huang, L., Human, J., Long, A., Newcomb, J., Patel, V.F., Saffran, D., Serafino, R., Schneider, S., Strathdee, C., Tang, J., Turci, S., White, R., Yu, V., Zhao, H., Wilson, C., Martin, M.W.
ACS Med Chem Lett
HeaderTransferase/Transferase Inhibitor
Released2012-10-08
Resolution1.800
CATH Insert Date02 Dec, 2012

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 31 Dec, 2012 Chopped
B 31 Dec, 2012 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4hgtA01 03 Jan, 2013 3.30.200.20 Assigned
4hgtA02 03 Jan, 2013 1.10.510.10 Assigned
4hgtB01 03 Jan, 2013 3.30.200.20 Assigned
4hgtB02 03 Jan, 2013 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta
P48730 KC1D_HUMAN Homo sapiens Casein kinase I isoform delta