PDB Information

PDB4GU6
MethodX-RAY DIFFRACTION
Host OrganismTrichoplusia ni
Gene SourceHomo sapiens
Primary Citation
Fragment-based discovery of new highly substituted 1H-pyrrolo[2,3-b]- and 3H-imidazolo[4,5-b]-pyridines as focal adhesion kinase inhibitors.
Heinrich, T., Seenisamy, J., Emmanuvel, L., Kulkarni, S.S., Bomke, J., Rohdich, F., Greiner, H., Esdar, C., Krier, M., Gradler, U., Musil, D.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2012-08-29
Resolution1.950
CATH Insert Date22 Sep, 2013

PDB Images (7)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 23 Sep, 2013 Chopped
B 23 Sep, 2013 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4gu6A01 25 Sep, 2013 3.30.200.20 Assigned
4gu6A02 25 Sep, 2013 1.10.510.10 Assigned
4gu6B01 25 Sep, 2013 3.30.200.20 Assigned
4gu6B02 25 Sep, 2013 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
Q05397 FAK1_HUMAN Homo sapiens Focal adhesion kinase 1
Q05397 FAK1_HUMAN Homo sapiens Focal adhesion kinase 1