PDB 4frs
PDB Information
PDB | 4FRS |
Method | X-RAY DIFFRACTION |
Host Organism | Escherichia coli |
Gene Source | Homo sapiens |
Primary Citation | Discovery of an Orally Available, Brain Penetrant BACE1 Inhibitor That Affords Robust CNS A(beta) Reduction
ACS Med Chem Lett
|
Header | Hydrolase/Hydrolase Inhibitor |
Released | 2012-06-26 |
Resolution | 1.700 |
CATH Insert Date | 04 Nov, 2012 |
PDB Images (7)
PDB Prints
PDB Chains (2)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 05 Nov, 2012 | Chopped |
B | 05 Nov, 2012 | Chopped |
CATH Domains (4)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4frsA01 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
4frsA02 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
4frsB01 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
4frsB02 | 10 Nov, 2012 | 2.40.70.10 | Assigned |
UniProtKB Entries (2)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P56817 | BACE1_HUMAN | Homo sapiens | Beta-secretase 1 |
P56817 | BACE1_HUMAN | Homo sapiens | Beta-secretase 1 |