PDB Information

PDB4F0E
MethodX-RAY DIFFRACTION
Host OrganismEscherichia coli
Gene SourceHomo sapiens
Primary Citation
Discovery of Ligands for ADP-Ribosyltransferases via Docking-Based Virtual Screening.
Andersson, C.D., Karlberg, T., Ekblad, T., Lindgren, A.E., Thorsell, A.G., Spjut, S., Uciechowska, U., Niemiec, M.S., Wittung-Stafshede, P., Weigelt, J., Elofsson, M., Schuler, H., Linusson, A.
J.Med.Chem.
HeaderTransferase/Transferase Inhibitor
Released2012-05-04
Resolution2.400
CATH Insert Date04 Nov, 2012

PDB Images (9)

PDB Prints

PDB Chains (4)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped
B 05 Nov, 2012 Chopped
C 05 Nov, 2012 Chopped
D 05 Nov, 2012 Chopped

CATH Domains (4)

Domain ID Date inserted into CATH Superfamily CATH Status
4f0eA00 10 Nov, 2012 3.90.228.10 Assigned
4f0eB00 10 Nov, 2012 3.90.228.10 Assigned
4f0eC00 10 Nov, 2012 3.90.228.10 Assigned
4f0eD00 10 Nov, 2012 3.90.228.10 Assigned

UniProtKB Entries (4)

Accession Gene ID Taxon Description
Q460N3 PAR15_HUMAN Homo sapiens Protein mono-ADP-ribosyltransferase PARP15
Q460N3 PAR15_HUMAN Homo sapiens Protein mono-ADP-ribosyltransferase PARP15
Q460N3 PAR15_HUMAN Homo sapiens Protein mono-ADP-ribosyltransferase PARP15
Q460N3 PAR15_HUMAN Homo sapiens Protein mono-ADP-ribosyltransferase PARP15