PDB 4e4l
PDB Information
PDB | 4E4L |
Method | X-RAY DIFFRACTION |
Host Organism | Spodoptera frugiperda |
Gene Source | Homo sapiens |
Primary Citation | Identification of Imidazo-Pyrrolopyridines as Novel and Potent JAK1 Inhibitors.
J.Med.Chem.
|
Header | Transferase/Transferase Inhibitor |
Released | 2012-03-13 |
Resolution | 2.000 |
CATH Insert Date | 03 Jun, 2012 |
PDB Images (13)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 03 Jun, 2012 | Chopped |
B | 03 Jun, 2012 | Chopped |
D | 03 Jun, 2012 | Chopped |
E | 03 Jun, 2012 | Chopped |
CATH Domains (8)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
4e4lA01 | 08 Jun, 2012 | 3.30.200.20 | Assigned |
4e4lA02 | 08 Jun, 2012 | 1.10.510.10 | Assigned |
4e4lB01 | 08 Jun, 2012 | 3.30.200.20 | Assigned |
4e4lB02 | 08 Jun, 2012 | 1.10.510.10 | Assigned |
4e4lD01 | 08 Jun, 2012 | 3.30.200.20 | Assigned |
4e4lD02 | 08 Jun, 2012 | 1.10.510.10 | Assigned |
4e4lE01 | 08 Jun, 2012 | 3.30.200.20 | Assigned |
4e4lE02 | 08 Jun, 2012 | 1.10.510.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
P23458 | JAK1_HUMAN | Homo sapiens | Tyrosine-protein kinase JAK1 |
P23458 | JAK1_HUMAN | Homo sapiens | Tyrosine-protein kinase JAK1 |
P23458 | JAK1_HUMAN | Homo sapiens | Tyrosine-protein kinase JAK1 |
P23458 | JAK1_HUMAN | Homo sapiens | Tyrosine-protein kinase JAK1 |