PDB Information

PDB4AZE
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Selectivity, Co-Crystal Structures and Neuroprotective Properties of Leucettines, a Family of Protein Kinase Inhibitors Derived from the Marine Sponge Alkaloid Leucettamine B.
Tahtouh, T., Elkins, J.M., Filippakopoulos, P., Soundararajan, M., Burgy, G., Durieu, E., Cochet, C., Schmid, R.S., Lo, D.C., Delhommel, F., Oberholzer, A., Laurence, P., Carreaux, F., Bazureau, J.P., Knapp, S., Meijer, L.
J.Med.Chem.
HeaderTransferase
Released2012-06-25
Resolution3.150
CATH Insert Date04 Nov, 2012

PDB Images (13)

PDB Prints

PDB Chains (6)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped
B 05 Nov, 2012 Chopped
C 05 Nov, 2012 Chopped
E 05 Nov, 2012 Rejected
F 05 Nov, 2012 Rejected
G 05 Nov, 2012 Rejected

CATH Domains (6)

Domain ID Date inserted into CATH Superfamily CATH Status
4azeA01 23 Jul, 2013 3.30.200.20 Assigned
4azeA02 23 Jul, 2013 1.10.510.10 Assigned
4azeB01 23 Jul, 2013 3.30.200.20 Assigned
4azeB02 23 Jul, 2013 1.10.510.10 Assigned
4azeC01 23 Jul, 2013 3.30.200.20 Assigned
4azeC02 23 Jul, 2013 1.10.510.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A
Q13627 DYR1A_HUMAN Homo sapiens Dual specificity tyrosine-phosphorylation-regulated kinase 1A