PDB Information

PDB4AWI
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
4-Phenyl-7-Azaindoles as Potent, Selective and Bioavailable Ikk2 Inhibitors Demonstrating Good in Vivo Efficacy.
Liddle, J., Bamborough, P., Barker, M.D., Campos, S., Chung, C., Cousins, R.P.C., Faulder, P., Heathcote, M.L., Hobbs, H., Holmes, D.S., Ioannou, C., Ramirez-Molina, C., Morse, M.A., Osborn, R., Payne, J.J., Pritchard, J.M., Rumsey, W.L., Tape, D.T., Vicentini, G., Whitworth, C., Williamson, R.A.
Bioorg.Med.Chem.Lett.
HeaderTransferase
Released2012-06-03
Resolution1.910
CATH Insert Date07 Jul, 2013

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 08 Jul, 2013 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
4awiA01 09 Aug, 2013 3.30.200.20 Assigned
4awiA02 09 Aug, 2013 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P45983 MK08_HUMAN Homo sapiens Mitogen-activated protein kinase 8