PDB Information

PDB4A9M
MethodX-RAY DIFFRACTION
Host OrganismESCHERICHIA COLI
Gene SourceHOMO SAPIENS
Primary Citation
Fragment-Based Discovery of Bromodomain Inhibitors Part 2: Optimization of Phenylisoxazole Sulfonamides.
Bamborough, P., Diallo, H., Goodacre, J.D., Gordon, L., Lewis, A., Seal, J.T., Wilson, D.M., Woodrow, M.D., Chung, C.W.
J.Med.Chem.
HeaderSignaling Protein
Released2011-11-26
Resolution2.060
CATH Insert Date12 Feb, 2012

PDB Images (7)

PDB Prints

PDB Chains (3)

Chain ID Date inserted into CATH CATH Status
A 13 Feb, 2012 Chopped
B 13 Feb, 2012 Chopped
C 13 Feb, 2012 Chopped

CATH Domains (3)

Domain ID Date inserted into CATH Superfamily CATH Status
4a9mA00 16 Feb, 2012 1.20.920.10 Assigned
4a9mB00 16 Feb, 2012 1.20.920.10 Assigned
4a9mC00 16 Feb, 2012 1.20.920.10 Assigned

UniProtKB Entries (3)

Accession Gene ID Taxon Description
P25440 BRD2_HUMAN Homo sapiens Bromodomain-containing protein 2
P25440 BRD2_HUMAN Homo sapiens Bromodomain-containing protein 2
P25440 BRD2_HUMAN Homo sapiens Bromodomain-containing protein 2
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