PDB Information

PDB3ZDI
MethodX-RAY DIFFRACTION
Host OrganismSPODOPTERA FRUGIPERDA
Gene SourceHOMO SAPIENS
Primary Citation
3,6-Diamino-4-(2-Halophenyl)-2-Benzoylthieno(2,3-B) Pyridine-5-Carbonitriles are Selective Inhibitors of Plasmodium Falciparum Glycogen Synthase Kinase-3 (Pfgsk-3)
Fugel, W., Oberholzer, A.E., Gschloessl, B., Dzikowski, R., Pressburger, N., Preu, L., Pearl, L.H., Baratte, B., Ratin, M., Okun, I., Doerig, C., Kruggel, S., Lemcke, T., Meijer, L., Kunick, C.
J.Med.Chem.
HeaderTransferase/Peptide
Released2012-11-27
Resolution2.650
CATH Insert Date13 Jan, 2013

PDB Images (5)

PDB Prints

PDB Chains (2)

Chain ID Date inserted into CATH CATH Status
A 14 Jan, 2013 Chopped
B 14 Jan, 2013 Rejected

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3zdiA01 18 Jan, 2013 3.30.200.20 Assigned
3zdiA02 18 Jan, 2013 1.10.510.10 Assigned

UniProtKB Entries (2)

Accession Gene ID Taxon Description
O15169 AXIN1_HUMAN Homo sapiens Axin-1
P49841 GSK3B_HUMAN Homo sapiens Glycogen synthase kinase-3 beta