PDB 3v8s
PDB Information
PDB | 3V8S |
Method | X-RAY DIFFRACTION |
Host Organism | Spodoptera frugiperda |
Gene Source | Homo sapiens |
Primary Citation | Fragment-based and structure-guided discovery and optimization of rho kinase inhibitors.
J.Med.Chem.
|
Header | Transferase/Transferase Inhibitor |
Released | 2011-12-23 |
Resolution | 2.290 |
CATH Insert Date | 12 Feb, 2012 |
PDB Images (13)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 13 Feb, 2012 | Chopped |
B | 13 Feb, 2012 | Chopped |
C | 13 Feb, 2012 | Chopped |
D | 13 Feb, 2012 | Chopped |
CATH Domains (8)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
3v8sA01 | 25 Apr, 2013 | 3.30.200.20 | Assigned |
3v8sA02 | 25 Apr, 2013 | 1.10.510.10 | Assigned |
3v8sB01 | 25 Apr, 2013 | 3.30.200.20 | Assigned |
3v8sB02 | 25 Apr, 2013 | 1.10.510.10 | Assigned |
3v8sC01 | 25 Apr, 2013 | 3.30.200.20 | Assigned |
3v8sC02 | 25 Apr, 2013 | 1.10.510.10 | Assigned |
3v8sD01 | 25 Apr, 2013 | 3.30.200.20 | Assigned |
3v8sD02 | 25 Apr, 2013 | 1.10.510.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q13464 | ROCK1_HUMAN | Homo sapiens | Rho-associated protein kinase 1 |
Q13464 | ROCK1_HUMAN | Homo sapiens | Rho-associated protein kinase 1 |
Q13464 | ROCK1_HUMAN | Homo sapiens | Rho-associated protein kinase 1 |
Q13464 | ROCK1_HUMAN | Homo sapiens | Rho-associated protein kinase 1 |