PDB 3v5l
PDB Information
PDB | 3V5L |
Method | X-RAY DIFFRACTION |
Host Organism | Spodoptera frugiperda |
Gene Source | Homo sapiens |
Primary Citation | X-ray crystallographic structure-based design of selective thienopyrazole inhibitors for interleukin-2-inducible tyrosine kinase.
Bioorg.Med.Chem.Lett.
|
Header | Transferase/Transferase Inhibitor |
Released | 2011-12-16 |
Resolution | 1.860 |
CATH Insert Date | 27 May, 2012 |
PDB Images (13)
PDB Prints
PDB Chains (4)
Chain ID | Date inserted into CATH | CATH Status |
---|---|---|
A | 28 May, 2012 | Chopped |
B | 28 May, 2012 | Chopped |
C | 28 May, 2012 | Chopped |
D | 28 May, 2012 | Chopped |
CATH Domains (8)
Domain ID | Date inserted into CATH | Superfamily | CATH Status |
---|---|---|---|
3v5lA01 | 08 Jun, 2012 | 3.30.200.20 | Assigned |
3v5lA02 | 08 Jun, 2012 | 1.10.510.10 | Assigned |
3v5lB01 | 08 Jun, 2012 | 3.30.200.20 | Assigned |
3v5lB02 | 08 Jun, 2012 | 1.10.510.10 | Assigned |
3v5lC01 | 08 Jun, 2012 | 3.30.200.20 | Assigned |
3v5lC02 | 08 Jun, 2012 | 1.10.510.10 | Assigned |
3v5lD01 | 08 Jun, 2012 | 3.30.200.20 | Assigned |
3v5lD02 | 08 Jun, 2012 | 1.10.510.10 | Assigned |
UniProtKB Entries (4)
Accession | Gene ID | Taxon | Description |
---|---|---|---|
Q08881 | ITK_HUMAN | Homo sapiens | Tyrosine-protein kinase ITK/TSK |
Q08881 | ITK_HUMAN | Homo sapiens | Tyrosine-protein kinase ITK/TSK |
Q08881 | ITK_HUMAN | Homo sapiens | Tyrosine-protein kinase ITK/TSK |
Q08881 | ITK_HUMAN | Homo sapiens | Tyrosine-protein kinase ITK/TSK |