PDB Information

PDB3UMW
MethodX-RAY DIFFRACTION
Host Organismcell-free protein synthesis
Gene SourceHomo sapiens
Primary Citation
Rational evolution of a novel type of potent and selective proviral integration site in Moloney murine leukemia virus kinase 1 (PIM1) inhibitor from a screening-hit compound.
Nakano, H., Saito, N., Parker, L.J., Tada, Y., Abe, M., Tsuganezawa, K., Yokoyama, S., Tanaka, A., Kojima, H., Okabe, T., Nagano, T.
J.Med.Chem.
HeaderTransferase/Inhibitor
Released2011-11-14
Resolution2.080
CATH Insert Date04 Nov, 2012

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 05 Nov, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3umwA01 10 Nov, 2012 3.30.200.20 Assigned
3umwA02 10 Nov, 2012 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
P11309 PIM1_HUMAN Homo sapiens Serine/threonine-protein kinase pim-1