PDB Information

PDB3U9N
MethodX-RAY DIFFRACTION
Host OrganismSpodoptera frugiperda
Gene SourceHomo sapiens
Primary Citation
Discovery of a Novel Series of CHK1 Kinase Inhibitors with Distinctive Hinge Binding Mode
Huang, X., Cheng, C.C., Fischmann, T.O., Duca, J.S., Yang, X., Richards, M., Shipps Jr., G.W.
ACS MED.CHEM.LETT.
HeaderTransferase/Transferase Inhibitor
Released2011-10-19
Resolution1.850
CATH Insert Date29 Jan, 2012

PDB Images (4)

PDB Prints

PDB Chains (1)

Chain ID Date inserted into CATH CATH Status
A 30 Jan, 2012 Chopped

CATH Domains (2)

Domain ID Date inserted into CATH Superfamily CATH Status
3u9nA01 02 Feb, 2012 3.30.200.20 Assigned
3u9nA02 02 Feb, 2012 1.10.510.10 Assigned

UniProtKB Entries (1)

Accession Gene ID Taxon Description
O14757 CHK1_HUMAN Homo sapiens Serine/threonine-protein kinase Chk1