Pyrazolopyridine Inhibitors of B-Raf(V600E). Part 1: The Development of Selective, Orally Bioavailable, and Efficacious Inhibitors.
Wenglowsky, S., Ren, L., Ahrendt, K.A., Laird, E.R., Aliagas, I., Alicke, B., Buckmelter, A.J., Choo, E.F., Dinkel, V., Feng, B., Gloor, S.L., Gould, S.E., Gross, S., Gunzner-Toste, J., Hansen, J.D., Hatzivassiliou, G., Liu, B., Malesky, K., Mathieu, S., Newhouse, B., Raddatz, N.J., Ran, Y., Rana, S., Randolph, N., Risom, T., Rudolph, J., Savage, S., Selby, L.T., Shrag, M., Song, K., Sturgis, H.L., Voegtli, W.C., Wen, Z., Willis, B.S., Woessner, R.D., Wu, W.I., Young, W.B., Grina, J.
ACS Med Chem Lett